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Recruiting NCT04546126

Positron Emission Tomography (PET) Imaging of Cholesterol Trafficking: Clinical Evaluation of [18F]FNP-59 in Normal Human Subjects (Groups 2, 3 & 4)

Early Phase I Interventional Radiotracer Hypertension Cholesterol

For patients and families

In plain language

An automatic summary of structured registry data. It is an orientation aid, not a substitute for the official protocol or a physician assessment.

What is being studied
The protocol lists: Dexamethasone (Group 2), Cosyntropin (Group 3), PET/CT Scan with FNP-59.
Who it may be relevant to
Registry conditions: Radiotracer, Hypertension, Cholesterol. Basic parameters: from 18 years · All.
What needs checking
Age, condition and sex are only basic indicators. Prior treatment, laboratory values and other mandatory requirements appear in the eligibility criteria below.
Where it takes place
United States
Next step
Save the trial, show it to the treating physician, and confirm current recruitment with the study center. Costs, documents and travel →

Overview

This study will evaluate the feasibility of using a sub-therapeutic dose of a fluorine-18 analogue of NP-59 (\[18F\]FNP-59) to image the adrenal gland. Some participants are healthy normal subjects but have undergone interventions to manipulate hormones while other participants have known adrenal pathology.

Detailed description

Groups 2 \& 3 used hormone manipulation using information gathered from Group 1 which identified radiation dosimetry and optimal uptake time.

Group 4 (added to the study later) includes participants with known adrenal pathology. They will not have study associated hormone manipulation.

All groups will be given a radio-tracer and PET/CT scans.

The researchers believe that a fluorine-18 analogue of NP-59, \[18F\]FNP-59, would greatly improve the imaging characteristics, by providing a PET imaging cholesterol analogue with significantly improved radiation dosimetry, and improved localization / sensitivity / specificity without concern of thyroid exposure.

Interventions

  • Drug Dexamethasone (Group 2)
    Participants will take 1 mg dexamethasone 2x a day for 3 days to suppress cortisol production.
  • Drug Cosyntropin (Group 3)
    Cosyntropin, 250 micro-gm will be administered IV. Five minutes following administration FNP-59 will be given. Following uptake of FNP-59 imaging will occur.
  • Combination product PET/CT Scan with FNP-59
    FNP-59, a radiotracer, is administered for PET/CT scans.

Primary outcome measures

  • Change in [18F]FNP-59 chemistry uptake as measured by the standardized uptake value (SUV) based gland segmentation [Time frame: Day 0, Day 4]
Secondary outcome measures (1)
  • PET/CT image uptake score as measured by investigator visual assessment for each volume of interest (VOI) [Time frame: Day 4]

Eligibility criteria

Inclusion Criteria (Groups 2 \& 3):

  • Participants without any known adrenal pathology as normal controls for undergoing endocrine manipulation

Exclusion Criteria (Groups 2 \& 3):

  • Pregnancy
  • Unable to do imaging
  • Body weight greater than 400 lbs (181 Kg)
  • Prisoners are not eligible
  • Subjects unable to provide own consent are not eligible
  • Current use of steroids, Oral contraceptives (OCP), spironolactone, estrogen, androgen, progesterone, Angiotensin-converting enzyme (ACE inhibitors)/ Angiotensin II receptor blockers (ARBs), or supplements that are hormone analogues.
  • Known adrenal pathology

Inclusion Criteria (Group 4):

  • Abnormal adrenal cortical hormone secretion

Exclusion Criteria (Group 4):

  • Pregnant

Criteria are shown verbatim from the registry (in English). Final eligibility is always assessed by the study center.

Healthy volunteers: Yes

Study design

Allocation
Non-randomized
Model
Parallel assignment
Masking
Open label
Primary purpose
Health services research

Study locations

United States · 2 centers
  • University of Michigan — Ann Arbor
  • BAMF Health, Inc. — Grand Rapids

Identifiers

NCT: NCT04546126 · HUM00179097b

Primary sources (government registries)

View this study on ClinicalTrials.gov ↗